Basic Peptide Information

DICL ID
DICL_Pep_00501
Ion Channel
Voltage-gated potassium channel subfamily KQT member 2/3
Peptide Function
Inhibitor
Gene Name
KCNQ2/KCNQ3

Activity Data (nM)

IC50
5000 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified

Sequence Information

Peptide Sequence
CNCKAPETALCARRCQQH
Peptide UniProt Accession
UniParc
UPI0000035420
Peptide Synonyms/Alias
[Apamin; Apamine; UNII-X644P85KUR; EINECS 246-182-7; C79H131N31O24S4; Ro 23-6721; X644P85KUR; NS00075519; Q417260]
Peptide Species
Apis mellifera (Honeybee)
Peptide Name
Apamin
CAS Number
24345-16-2

Experimental Conditions

pH
pH 7.4
Holding Potential (mV)
−90 mV
Temperature
18–22 °C
Test Method
Patch-clamping
Test Species
Xenopus laevis oocyte

Binding Information

Binding Site
Not specified
Binding Site Residue
Not specified

Ion Channel Information

Gene Abbreviation (ABB)
VGKCs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)

References & Disease Information

Disease
Not specified
PubChem CID
URL
Not available
PMID
Patent
Not available